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英文名 :Matrix Metalloproteinase-13 (MMP-13) fluorometric drug discovery kit
规格 :96wells
基质金属蛋白酶-13(MMP-13)的药物drug discovery kitMatrix Metalloproteinase-13 (MMP-13) fluorometric drug discovery kit
A QuantiZyme™ Assay System. The MMP-13 Fluorometric (also known as fluorimetric) Drug Discovery Kit is a complete assay system designed to screen inhibitors of matrix metalloproteinase-13 (MMP-13, collagenase-3) using a quenched fluorogenic peptide: OMNIMMP® fluorogenic substrate Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH. Mca fluorescence is quenched by the Dpa group until cleavage by MMPs at the Gly-Leu bond separates the two moieties. The assays are performed in a convenient 96-well microplate format. The kit is useful to screen inhibitors of MMP-13, a potential therapeutic target. Included are active enzyme, assay buffer, a prototypic control inhibitor (NNGH3), and a detailed instruction booklet.
Product Specification
Alternative Name: | Collagenase-3 |
Applications: | Fluorescent detection, HTS Activity assay |
Shipping: | Shipped on Dry Ice |
Long Term Storage: | -80°C |
Kit/Set Contains: | MMP-13 enzyme (human) (recombinant), substrate, calibration standard, inhibitor, assay buffer, 96-well white microplate. |
UniProt ID: | P45452 |
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