MCE 的所有产品仅用作科学研究或药证申报，我们不为任何个人用途提供产品和服务。

Src Inhibitor 1

CAS No. : 179248-59-0

MCE 国际站：Src Inhibitor 1

产品活性：Src Inhibitor 1是高效选择性的，ATP-竞争性的双位点Src酪氨酸激酶抑制剂，对Src和Lck的IC₅₀值分别为44 nM和88 nM。

研究领域：Protein Tyrosine Kinase/RTK

作用靶点：Src

In Vitro: Src Inhibitor 1 is competitive with both ATP and peptide binding sites of the kinase. The IC₅₀ values are 44 and 88 nM for Src and Lck, respectively. Src Inhibitor 1 is found to be a potent inhibitor of Src (IC₅₀=0.18 μM), but also inhibited other Src family members, such as Lck, Csk and Yes with similar potency to Src, and RIP2 (IC₅₀=0.026 μM) with even greater potency. In addition, it inhibited CHK2 with similar potency to Src, and Aurora B with slightly lower potency.

相关产品：Bioactive Compound Library Plus  |  Kinase Inhibitor Library  |  Protein Tyrosine Kinase Compound Library  |  Anti-Cancer Compound Library  |  Reprogramming Compound Library  |  Anti-Pancreatic Cancer Compound Library  |  Angiogenesis-Related Compound Library  |  Targeted Diversity Library  |  Anti-Prostate Cancer Compound Library  |  Anti-Pulmonary Fibrosis Compound Library  |  Heterocyclic Compound Library  |  Pain-Related Compound Library  |  Membrane Protein-targeted Compound Library  |  Highly Selective Inhibitors Library  |  Dasatinib  |  Ponatinib  |  Saracatinib  |  Bosutinib  |  PP2  |  Rebastinib  |  Masitinib  |  A 419259 trihydrochloride  |  WH-4-023  |  Tirbanibulin  |  Bafetinib  |  PP1  |  SU6656  |  eCF506  |  Lck Inhibitor  |  Pelitinib  |  1-NM-PP1  |  SM1-71  |  Scutellarein  |  1-Naphthyl PP1  |  CH6953755  |  PP121  |  TL02-59  |  RK-24466  |  PD173955  |  Tolimidone  |  A-770041  |  ENMD-2076

热门产品线：重组蛋白  |  化合物库  |  天然产物  |  荧光染料  |  PROTAC  |  同位素标记物

Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  |  Natural Products  |  Dye Reagents  |  PROTAC  |  Isotope-Labeled Compounds