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保存条件 :4°C, sealed storage, away from moisture
英文名 :CVT 303-dd<sub>8</sub> dihydrochloride; RS 43285-d<sub>8</sub>
库存 :货期:1-2天
供应商 :MedChemExpress LLC
CAS号 :1219802-60-4
规格 :1 mg
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Ranolazine-d8 dihydrochloride
CAS No. : 1219802-60-4
MCE 国际站:Ranolazine-d8 dihydrochloride
产品活性:Ranolazine-d8 (dihydrochloride) 是 Ranolazine dihydrochloride 的氘代物。Ranolazine dihydrochloride (CVT 303 dihydrochloride) 是一种抗心绞痛和抗缺血剂,可通过抑制内向钠电流的后期作用 (对 INa 和 IKr 的 IC50 值分别为 6 μM 和 12 μM) 来发挥功效,而不会影响心率或血压。Ranolazine dihydrochloride 还是脂肪酸氧化的部分抑制剂。
研究领域:Membrane Transporter/Ion Channel | Neuronal Signaling | Autophagy
作用靶点:Calcium Channel | Sodium Channel | Autophagy
In Vitro: Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs.
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